MW 448.39 g/mol, Purity >99%. Partial dopamine D₂ agonist. Ki (nM) values are 265 (D₁), 0.34 (D₂), 0.8 (D₃), 44 (D₄), 1.7 (5-HT₁A), 3.4 (5-HT₂A), 15 (5-HT₂C), 214 (5-HT₆), 39 (5-HT₇), 57 (α₁), 791 (α₂), 61 (H₁) and >1000 (M₁). Antipsychotic and antidepressant activity. Centrally active following oral administration.
The product is subject to the following: Abcam Restricted Use Statement